5IKW
Crystal Structure of BMP-2-inducible kinase in complex with an Indazole inhibitor
Summary for 5IKW
Entry DOI | 10.2210/pdb5ikw/pdb |
Descriptor | BMP-2-inducible protein kinase, N-(6-{3-[(cyclopropylsulfonyl)amino]phenyl}-1H-indazol-3-yl)cyclopropanecarboxamide (3 entities in total) |
Functional Keywords | transferase, protein kinase domain, structural genomics, structural genomics consortium, sgc, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus : Q9NSY1 |
Total number of polymer chains | 1 |
Total formula weight | 35187.50 |
Authors | Counago, R.M.,Sorrell, F.J.,Krojer, T.,Savitsky, P.,Elkins, J.M.,Axtman, A.,Drewry, D.,Wells, C.,Zhang, C.,Zuercher, W.,Willson, T.M.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Arruda, P.,Gileadi, O.,Structural Genomics Consortium (SGC) (deposition date: 2016-03-04, release date: 2016-06-29, Last modification date: 2024-01-10) |
Primary citation | Counago, R.M.,Sorrell, F.J.,Krojer, T.,Savitsky, P.,Elkins, J.M.,Axtman, A.,Drewry, D.,Wells, C.,Zhang, C.,Zuercher, W.,Willson, T.M.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Arruda, P.,Gileadi, O.,Structural Genomics Consortium (SGC) Crystal Structure of BMP-2-inducible kinase in complex with a 3-acylaminoindazole inhibitor GSK3236425A To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.41 Å) |
Structure validation
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