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5IBK

Skp1-F-box in complex with a ubiquitin variant

Summary for 5IBK
Entry DOI10.2210/pdb5ibk/pdb
DescriptorS-phase kinase-associated protein 1,S-phase kinase-associated protein 1, F-box/WD repeat-containing protein 7, Polyubiquitin-B, ... (4 entities in total)
Functional Keywordsphage display, scf inhibitors, fbxw7, fbxw11, ?-trcp, ubiquitin, protein binding
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains6
Total formula weight66612.28
Authors
Orlicky, S.,Sicheri, F. (deposition date: 2016-02-22, release date: 2016-03-30, Last modification date: 2023-09-27)
Primary citationGorelik, M.,Orlicky, S.,Sartori, M.A.,Tang, X.,Marcon, E.,Kurinov, I.,Greenblatt, J.F.,Tyers, M.,Moffat, J.,Sicheri, F.,Sidhu, S.S.
Inhibition of SCF ubiquitin ligases by engineered ubiquitin variants that target the Cul1 binding site on the Skp1-F-box interface.
Proc.Natl.Acad.Sci.USA, 113:3527-3532, 2016
Cited by
PubMed: 26976582
DOI: 10.1073/pnas.1519389113
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.503 Å)
Structure validation

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