Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4X9W

PLK-1 polo-box domain in complex with Bioactive Imidazolium-containing phosphopeptide macrocycle 4C

Summary for 4X9W
Entry DOI10.2210/pdb4x9w/pdb
Related4X9R
DescriptorSerine/threonine-protein kinase PLK1, Macrocyclic phosphopeptide 4C (3 entities in total)
Functional Keywordstransferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (Human)
More
Cellular locationNucleus: P53350
Total number of polymer chains2
Total formula weight28194.24
Authors
Grant, R.A.,Qian, W.-J.,Yaffe, M.B.,Burke, T.R. (deposition date: 2014-12-11, release date: 2015-07-29, Last modification date: 2023-11-15)
Primary citationQian, W.J.,Park, J.E.,Grant, R.,Lai, C.C.,Kelley, J.A.,Yaffe, M.B.,Lee, K.S.,Burke, T.R.
Neighbor-directed histidine N ( tau )-alkylation: A route to imidazolium-containing phosphopeptide macrocycles.
Biopolymers, 104:663-673, 2015
Cited by
PubMed: 26152807
DOI: 10.1002/bip.22698
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.798 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon