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4UXN

LSD1(KDM1A)-CoREST in complex with Z-Pro derivative of MC2580

Summary for 4UXN
Entry DOI10.2210/pdb4uxn/pdb
DescriptorLYSINE-SPECIFIC HISTONE DEMETHYLASE 1A, REST COREPRESSOR 1, FLAVIN-ADENINE DINUCLEOTIDE, ... (4 entities in total)
Functional Keywordsoxidoreductase, covalent inhibitor, tranylcypromine
Biological sourceHOMO SAPIENS (HUMAN)
More
Total number of polymer chains2
Total formula weight147279.40
Authors
Rodriguez, V.,Valente, S.,Stazi, G.,Lucidi, A.,Mercurio, C.,Vianello, P.,Ciossani, G.,Mattevi, A.,Botrugno, O.A.,Dessanti, P.,Minucci, S.,Varasi, M.,Mai, A. (deposition date: 2014-08-27, release date: 2015-02-25, Last modification date: 2024-01-10)
Primary citationRodriguez, V.,Valente, S.,Rovida, S.,Rotili, D.,Stazi, G.,Lucidi, A.,Ciossani, G.,Mattevi, A.,Botrugno, O.A.,Dessanti, P.,Mercurio, C.,Vianello, P.,Minucci, S.,Varasi, M.,Mai, A.
Pyrrole- and Indole-Containing Tranylcypromine Derivatives as Novel Lysine-Specific Demethylase 1 Inhibitors Active on Cancer Cells
Chemmedchem, 6:665-670, 2015
Cited by
DOI: 10.1039/C4MD00507D
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.85 Å)
Structure validation

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