Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4EH2

Human p38 MAP kinase in complex with NP-F1 and RL87

Summary for 4EH2
Entry DOI10.2210/pdb4eh2/pdb
Related4EH3 4EH4 4EH5 4EH6 4EH7 4EH8 4EH9
DescriptorMitogen-activated protein kinase 14, N~4~-cyclopropyl-2-phenylquinazoline-4,7-diamine, 3-phenylquinazolin-4(3H)-one, ... (4 entities in total)
Functional Keywordsmap kinase insert, kinase-ligand complex, np-fragment, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm: Q16539
Total number of polymer chains1
Total formula weight41767.63
Authors
Over, B.,Gruetter, C.,Waldmann, H.,Rauh, D. (deposition date: 2012-04-02, release date: 2012-12-05, Last modification date: 2023-09-13)
Primary citationOver, B.,Wetzel, S.,Grutter, C.,Nakai, Y.,Renner, S.,Rauh, D.,Waldmann, H.
Natural-product-derived fragments for fragment-based ligand discovery.
Nat Chem, 5:21-28, 2012
Cited by
PubMed: 23247173
DOI: 10.1038/nchem.1506
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon