4BPI
Mcl-1 bound to alpha beta Puma BH3 peptide 2
Summary for 4BPI
Entry DOI | 10.2210/pdb4bpi/pdb |
Related | 4BPJ 4BPK |
Descriptor | FUSION PROTEIN CONSISTING OF INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1 HOMOLOG, ALPHA BETA BH3PEPTIDE, CADMIUM ION, ... (4 entities in total) |
Functional Keywords | apoptosis, chimera, bim |
Biological source | MUS MUSCULUS (HOUSE MOUSE) More |
Total number of polymer chains | 2 |
Total formula weight | 21025.15 |
Authors | Smith, B.J.,Lee, E.F.,Checco, J.W.,Gellman, S.H.,Fairlie, W.D. (deposition date: 2013-05-27, release date: 2014-04-09, Last modification date: 2023-12-20) |
Primary citation | Smith, B.J.,Lee, E.F.,Checco, J.W.,Evangelista, M.,Gellman, S.H.,Fairlie, W.D. Structure-Guided Rational Design of Alpha/Beta-Peptide Foldamers with High Affinity for Bcl-2 Family Prosurvival Proteins. Chembiochem, 14:1564-, 2013 Cited by PubMed: 23929624DOI: 10.1002/CBIC.201300351 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.982 Å) |
Structure validation
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