Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4AZ0

crystal structure of cathepsin a, complexed with 8a.

Summary for 4AZ0
Entry DOI10.2210/pdb4az0/pdb
Related1IVY 4AZ3
DescriptorLYSOSOMAL PROTECTIVE PROTEIN 32 KDA CHAIN, LYSOSOMAL PROTECTIVE PROTEIN 20 KDA CHAIN, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (6 entities in total)
Functional Keywordshydrolase, drug discovery, cardiovascular drug
Biological sourceHOMO SAPIENS (HUMAN)
More
Total number of polymer chains2
Total formula weight53754.11
Authors
Primary citationRuf, S.,Buning, C.,Schreuder, H.,Horstick, G.,Linz, W.,Olpp, T.,Pernerstorfer, J.,Hiss, K.,Kroll, K.,Kannt, A.,Kohlmann, M.,Linz, D.,Hubschle, T.,Rutten, H.,Wirth, K.,Schmidt, T.,Sadowski, T.
Novel Beta-Amino Acid Derivatives as Inhibitors of Cathepsin A.
J.Med.Chem., 55:7636-, 2012
Cited by
PubMed: 22861813
DOI: 10.1021/JM300663N
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.17 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon