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4ANS

Structure of L1196M,G1269A Double Mutant Anaplastic Lymphoma Kinase in Complex with Crizotinib

Summary for 4ANS
Entry DOI10.2210/pdb4ans/pdb
Related4ANL 4ANQ 4AOI
DescriptorALK TYROSINE KINASE RECEPTOR, 3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)pyridin-2-amine (3 entities in total)
Functional Keywordstransferase
Biological sourceHOMO SAPIENS (HUMAN)
Total number of polymer chains1
Total formula weight39078.53
Authors
McTigue, M.,Deng, Y.,Liu, W.,Brooun, A. (deposition date: 2012-03-22, release date: 2013-03-27, Last modification date: 2023-12-20)
Primary citationMctigue, M.,Deng, Y.,Liu, W.,Brooun, A.
Structure of L1196M,G1269A Double Mutant Anaplastic Lymphoma Kinase in Complex with Crizotinib
To be Published,
Experimental method
X-RAY DIFFRACTION (1.85 Å)
Structure validation

217705

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