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4A07

Human PDK1 Kinase Domain in Complex with Allosteric Activator PS171 Bound to the PIF-Pocket

Summary for 4A07
Entry DOI10.2210/pdb4a07/pdb
Related1H1W 1OKY 1OKZ 1UU3 1UU7 1UU8 1UU9 1UVR 1W1D 1W1G 1W1H 1Z5M 2BIY 2VKI 2XCH 2XCK 4A06
Descriptor3-PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE 1, ADENOSINE-5'-TRIPHOSPHATE, (3S)-3-(4-CHLOROPHENYL)-4-(5,7-DICHLORO-1H-BENZIMIDAZOL-2-YL)BUTANOIC ACID, ... (6 entities in total)
Functional Keywordstransferase, allosteric site
Biological sourceHOMO SAPIENS (HUMAN)
Cellular locationCytoplasm: O15530
Total number of polymer chains1
Total formula weight36900.69
Authors
Schulze, J.O.,Lopez-Garcia, L.A.,Froehner, W.,Zhang, H.,Navratil, J.,Hindie, V.,Zeuzem, S.,Alzari, P.M.,Neimanis, S.,Engel, M.,Biondi, R.M. (deposition date: 2011-09-08, release date: 2011-12-07, Last modification date: 2023-12-20)
Primary citationLopez-Garcia, L.A.,Schulze, J.O.,Frohner, W.,Zhang, H.,Suss, E.,Weber, N.,Navratil, J.,Amon, S.,Hindie, V.,Zeuzem, S.,Jorgensen, T.J.,Alzari, P.M.,Neimanis, S.,Engel, M.,Biondi, R.M.
Allosteric Regulation of Protein Kinase Pkczeta by the N-Terminal C1 Domain and Small Compounds to the Pif-Pocket.
Chem.Biol., 18:1463-, 2011
Cited by
PubMed: 22118680
DOI: 10.1016/J.CHEMBIOL.2011.08.010
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.85 Å)
Structure validation

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