Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3U9Y

Crystal structure of human tankyrase 2 catalytic domain in complex with olaparib

Summary for 3U9Y
Entry DOI10.2210/pdb3u9y/pdb
Related3U9H 3UA9
DescriptorTankyrase-2, ZINC ION, SULFATE ION, ... (6 entities in total)
Functional Keywordsprotein-ligand complex, diphtheria toxin like fold, adp-ribosylation, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight28083.86
Authors
Narwal, M.,Lehtio, L. (deposition date: 2011-10-20, release date: 2012-01-25, Last modification date: 2023-09-13)
Primary citationNarwal, M.,Venkannagari, H.,Lehtio, L.
Structural basis of selective inhibition of human tankyrases.
J.Med.Chem., 55:1360-1367, 2012
Cited by
PubMed: 22233320
DOI: 10.1021/jm201510p
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon