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3MVJ

Human cyclic AMP-dependent protein kinase PKA inhibitor complex

Summary for 3MVJ
Entry DOI10.2210/pdb3mvj/pdb
Related3MV5 3MVH
DescriptorcAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha, (3R)-1-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine, ... (4 entities in total)
Functional Keywordskinase inhibitor, transferase
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm. Isoform 2: Cell projection, cilium, flagellum : P17612
Total number of polymer chains6
Total formula weight136053.52
Authors
Pandit, J.,Vajdos, F. (deposition date: 2010-05-04, release date: 2010-06-02, Last modification date: 2017-11-08)
Primary citationFreeman-Cook, K.D.,Autry, C.,Borzillo, G.,Gordon, D.,Barbacci-Tobin, E.,Bernardo, V.,Briere, D.,Clark, T.,Corbett, M.,Jakubczak, J.,Kakar, S.,Knauth, E.,Lippa, B.,Luzzio, M.J.,Mansour, M.,Martinelli, G.,Marx, M.,Nelson, K.,Pandit, J.,Rajamohan, F.,Robinson, S.,Subramanyam, C.,Wei, L.,Wythes, M.,Morris, J.
Design of selective, ATP-competitive inhibitors of Akt.
J.Med.Chem., 53:4615-4622, 2010
Cited by
PubMed: 20481595
DOI: 10.1021/jm1003842
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.49 Å)
Structure validation

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