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3G0B

Crystal structure of dipeptidyl peptidase IV in complex with TAK-322

3G0B の概要
エントリーDOI10.2210/pdb3g0b/pdb
関連するPDBエントリー3G0C 3G0D 3G0G
分子名称Dipeptidyl peptidase 4, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... (5 entities in total)
機能のキーワードprotease and 8-bladed beta-propeller domain, aminopeptidase, cell membrane, glycoprotein, hydrolase, membrane, protease, secreted, serine protease, signal-anchor, transmembrane, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
由来する生物種Homo sapiens (Human)
タンパク質・核酸の鎖数4
化学式量合計351617.09
構造登録者
主引用文献Zhang, Z.,Wallace, M.B.,Feng, J.,Stafford, J.A.,Skene, R.J.,Shi, L.,Lee, B.,Aertgeerts, K.,Jennings, A.,Xu, R.,Kassel, D.B.,Kaldor, S.W.,Navre, M.,Webb, D.R.,Gwaltney, S.L.
Design and Synthesis of Pyrimidinone and Pyrimidinedione Inhibitors of Dipeptidyl Peptidase IV.
J.Med.Chem., 54:510-524, 2011
Cited by
PubMed: 21186796
DOI: 10.1021/jm101016w
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (2.25 Å)
構造検証レポート
Validation report summary of 3g0b
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-03-27に公開中

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