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3E3B

Crystal structure of catalytic subunit of human protein kinase CK2alpha prime with a potent indazole-derivative inhibitor

Summary for 3E3B
Entry DOI10.2210/pdb3e3b/pdb
DescriptorCasein kinase II subunit alpha', [1-(6-{6-[(1-methylethyl)amino]-1H-indazol-1-yl}pyrazin-2-yl)-1H-pyrrol-3-yl]acetic acid (3 entities in total)
Functional Keywordscasein kinase 2, ck2alpha prime, ck2alpha inhibitor, selective kinase inhibitor, atp-binding, kinase, nucleotide-binding, polymorphism, serine/threonine-protein kinase, transferase, wnt signaling pathway
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight40536.40
Authors
Kinoshita, T.,Nakaniwa, T.,Tada, T. (deposition date: 2008-08-07, release date: 2009-03-03, Last modification date: 2023-11-01)
Primary citationNakaniwa, T.,Kinoshita, T.,Sekiguchi, Y.,Tada, T.,Nakanishi, I.,Kitaura, K.,Suzuki, Y.,Ohno, H.,Hirasawa, A.,Tsujimoto, G.
Structure of human protein kinase CK2alpha2 with a potent indazole-derivative inhibitor
Acta Crystallogr.,Sect.F, 65:75-79, 2009
Cited by
PubMed: 19193990
DOI: 10.1107/S1744309108043194
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3.2 Å)
Structure validation

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