Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3DJ7

Crystal structure of the mouse Aurora-A catalytic domain (Asn186->Gly, Lys240->Arg, Met302->Leu) in complex with Compound 130.

Summary for 3DJ7
Entry DOI10.2210/pdb3dj7/pdb
Related2c6d 3D2I 3D2K 3DJ5 3DJ6 3d14 3d15
Descriptorserine/threonine kinase 6, 1-(5-{2-[(6-amino-5-bromopyrimidin-4-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]urea (3 entities in total)
Functional Keywordsaurora a, small-molecule inhibitor, fragment-based drug discovery, kinase, transferase
Biological sourceMus musculus (mouse)
Total number of polymer chains1
Total formula weight32051.49
Authors
Elling, R.A.,Yang, W.,Erlanson, D.A.,Tangonan, B.T.,Hansen, S.K.,Romanowski, M.J. (deposition date: 2008-06-22, release date: 2009-05-05, Last modification date: 2023-08-30)
Primary citationElling, R.A.,Yang, W.,Erlanson, D.A.,Tangonan, B.T.,Hansen, S.K.,Romanowski, M.J.
New fragment-based drug discovery
To be Published,
Experimental method
X-RAY DIFFRACTION (2.8 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon