Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3C50

Crystal Structure of G protein coupled receptor kinase 1 bound to ADP and magnesium chloride at 2.6A

Summary for 3C50
Entry DOI10.2210/pdb3c50/pdb
Related3C4W 3C4X 3C4Y 3C4Z 3C51
DescriptorRhodopsin kinase, MAGNESIUM ION, CHLORIDE ION, ... (6 entities in total)
Functional Keywordsser/thr kinase, rgs homology domain, g protein coupled receptor kinase, grk, grk1, rhodopsin kinase, p-loop, autophosphorylation, adp, atp-binding, lipoprotein, membrane, methylation, nucleotide-binding, phosphoprotein, prenylation, serine/threonine-protein kinase, transferase
Biological sourceBos taurus (cattle)
Cellular locationMembrane; Lipid-anchor: P28327
Total number of polymer chains2
Total formula weight124290.35
Authors
Singh, P.,Tesmer, J.J.G. (deposition date: 2008-01-30, release date: 2008-03-11, Last modification date: 2023-08-30)
Primary citationSingh, P.,Wang, B.,Maeda, T.,Palczewski, K.,Tesmer, J.J.
Structures of rhodopsin kinase in different ligand states reveal key elements involved in G protein-coupled receptor kinase activation.
J.Biol.Chem., 283:14053-14062, 2008
Cited by
PubMed: 18339619
DOI: 10.1074/jbc.M708974200
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.6 Å)
Structure validation

218500

PDB entries from 2024-04-17

PDB statisticsPDBj update infoContact PDBjnumon