2W4O
Crystal structure of Human CAMK4 in complex with 4-Amino(sulfamoyl- phenylamino)-triazole-carbothioic acid (2,6-difluoro-phenyl)-amide)
Summary for 2W4O
Entry DOI | 10.2210/pdb2w4o/pdb |
Descriptor | CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE IV, 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE (3 entities in total) |
Functional Keywords | calmodulin-binding, nucleotide-binding, serine/threonine-protein kinase, atp-binding, phosphoprotein, kinase, nucleus, transferase |
Biological source | HOMO SAPIENS (HUMAN) |
Cellular location | Cytoplasm: Q16566 |
Total number of polymer chains | 1 |
Total formula weight | 39751.72 |
Authors | Muniz, J.R.C.,Rellos, P.,Gileadi, O.,Fedorov, O.,Filippakopoulos, P.,Salah, E.,Pike, A.,Phillips, C.,Niesen, F.,Shrestha, L.,Burgess-Brown, N.,Bullock, A.,Berridge, G.,von Delft, F.,Edwards, A.M.,Bountra, C.,Arrowsmith, C.H.,Weigelt, J.,Knapp, S. (deposition date: 2008-11-28, release date: 2009-01-20, Last modification date: 2024-02-07) |
Primary citation | Muniz, J.R.C.,Rellos, P.,Gileadi, O.,Fedorov, O.,Filippakopoulos, P.,Salah, E.,Pike, A.,Phillips, C.,Niesen, F.,Shrestha, L.,Burgess-Brown, N.,Bullock, A.,Berridge, G.,von Delft, F.,Edwards, A.M.,Bountra, C.,Arrowsmith, C.H.,Weigelt, J.,Knapp, S. Crystal Structure of Human Camk4 in Complex with 4-Amino(Sulfamoyl-Phenylamino)-Triazole- Carbothioic Acid (2,6-Difluoro-Phenyl)-Amide) To be Published, |
Experimental method | X-RAY DIFFRACTION (2.17 Å) |
Structure validation
Download full validation report