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2W4O

Crystal structure of Human CAMK4 in complex with 4-Amino(sulfamoyl- phenylamino)-triazole-carbothioic acid (2,6-difluoro-phenyl)-amide)

Summary for 2W4O
Entry DOI10.2210/pdb2w4o/pdb
DescriptorCALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE IV, 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE (3 entities in total)
Functional Keywordscalmodulin-binding, nucleotide-binding, serine/threonine-protein kinase, atp-binding, phosphoprotein, kinase, nucleus, transferase
Biological sourceHOMO SAPIENS (HUMAN)
Cellular locationCytoplasm: Q16566
Total number of polymer chains1
Total formula weight39751.72
Authors
Primary citationMuniz, J.R.C.,Rellos, P.,Gileadi, O.,Fedorov, O.,Filippakopoulos, P.,Salah, E.,Pike, A.,Phillips, C.,Niesen, F.,Shrestha, L.,Burgess-Brown, N.,Bullock, A.,Berridge, G.,von Delft, F.,Edwards, A.M.,Bountra, C.,Arrowsmith, C.H.,Weigelt, J.,Knapp, S.
Crystal Structure of Human Camk4 in Complex with 4-Amino(Sulfamoyl-Phenylamino)-Triazole- Carbothioic Acid (2,6-Difluoro-Phenyl)-Amide)
To be Published,
Experimental method
X-RAY DIFFRACTION (2.17 Å)
Structure validation

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