2PIV
Androgen receptor with small molecule
Summary for 2PIV
| Entry DOI | 10.2210/pdb2piv/pdb |
| Related | 2PIN 2PIO 2PIP 2PIQ 2PIR 2PIT 2PIU 2PIW 2PIX 2PKL |
| Descriptor | Androgen receptor, SULFATE ION, 5-ALPHA-DIHYDROTESTOSTERONE, ... (5 entities in total) |
| Functional Keywords | androgen receptor inhibitor coactivator binding, hormone receptor |
| Biological source | Homo sapiens (human) |
| Cellular location | Nucleus : P10275 |
| Total number of polymer chains | 1 |
| Total formula weight | 30314.82 |
| Authors | Estebanez-Perpina, E.,Arnold, A.A.,Baxter, J.D.,Webb, P.,Guy, R.K.,Fletterick, K.R. (deposition date: 2007-04-13, release date: 2007-09-25, Last modification date: 2023-11-15) |
| Primary citation | Estebanez-Perpina, E.,Arnold, L.A.,Arnold, A.A.,Nguyen, P.,Rodrigues, E.D.,Mar, E.,Bateman, R.,Pallai, P.,Shokat, K.M.,Baxter, J.D.,Guy, R.K.,Webb, P.,Fletterick, R.J. A surface on the androgen receptor that allosterically regulates coactivator binding. Proc.Natl.Acad.Sci.Usa, 104:16074-16079, 2007 Cited by PubMed: 17911242DOI: 10.1073/pnas.0708036104 PDB entries with the same primary citation |
| Experimental method | X-RAY DIFFRACTION (1.95 Å) |
Structure validation
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