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2PIU

Androgen receptor LBD with small molecule

Summary for 2PIU
Entry DOI10.2210/pdb2piu/pdb
Related2PIN 2PIO 2PIP 2PIQ 2PIR 2PIT 2PIV 2PIW 2PIX 2PKL
DescriptorAndrogen receptor, 5-ALPHA-DIHYDROTESTOSTERONE, [4-(4-HYDROXY-3-IODO-PHENOXY)-3,5-DIIODO-PHENYL]-ACETIC ACID, ... (4 entities in total)
Functional Keywordsandrogen receptor inhibitors coactivator binding af-2, hormone receptor
Biological sourceHomo sapiens (human)
Cellular locationNucleus : P10275
Total number of polymer chains1
Total formula weight30811.64
Authors
Estebanez-Perpina, E.,Arnold, A.A.,Baxter, J.D.,Webb, P.,Guy, R.K.,Fletterick, K.R. (deposition date: 2007-04-13, release date: 2007-09-25, Last modification date: 2024-02-21)
Primary citationEstebanez-Perpina, E.,Arnold, L.A.,Arnold, A.A.,Nguyen, P.,Rodrigues, E.D.,Mar, E.,Bateman, R.,Pallai, P.,Shokat, K.M.,Baxter, J.D.,Guy, R.K.,Webb, P.,Fletterick, R.J.
A surface on the androgen receptor that allosterically regulates coactivator binding.
Proc.Natl.Acad.Sci.Usa, 104:16074-16079, 2007
Cited by
PubMed: 17911242
DOI: 10.1073/pnas.0708036104
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.12 Å)
Structure validation

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