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2OVM

Progesterone Receptor with Bound Asoprisnil and a Peptide from the Co-Repressor NCoR

Summary for 2OVM
Entry DOI10.2210/pdb2ovm/pdb
Related1A28 2OVH
DescriptorProgesterone receptor, NCoR, 4-[(11BETA,17BETA)-17-METHOXY-17-(METHOXYMETHYL)-3-OXOESTRA-4,9-DIEN-11-YL]BENZALDEHYDE OXIME, ... (4 entities in total)
Functional Keywordsprogesterone receptor, pr, nuclear receptor, steroid receptor, co-repressor, asoprisnil, ncor, transcription
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight32654.21
Authors
Madauss, K.P.,Deng, S.-J.,Short, S.A.,Stewart, E.L.,Williams, S.P. (deposition date: 2007-02-14, release date: 2007-03-20, Last modification date: 2023-08-30)
Primary citationMadauss, K.P.,Grygielko, E.T.,Deng, S.J.,Sulpizio, A.C.,Stanley, T.B.,Wu, C.,Short, S.A.,Thompson, S.K.,Stewart, E.L.,Laping, N.J.,Williams, S.P.,Bray, J.D.
A structural and in vitro characterization of asoprisnil: a selective progesterone receptor modulator.
Mol.Endocrinol., 21:1066-1081, 2007
Cited by
PubMed: 17356170
DOI: 10.1210/me.2006-0524
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.6 Å)
Structure validation

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