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2IZR

Structure of casein kinase gamma 3 in complex with inhibitor

Summary for 2IZR
Entry DOI10.2210/pdb2izr/pdb
Related2CHL 2IZS 2IZT 2IZU
DescriptorCASEIN KINASE I ISOFORM GAMMA-3, {(2Z)-4-AMINO-2-[(4-METHOXYPHENYL)IMINO]-2,3-DIHYDRO-1,3-THIAZOL-5-YL}(4-METHOXYPHENYL)METHANONE, MAGNESIUM ION, ... (6 entities in total)
Functional Keywordsserine/threonine-protein kinase, kinase, transferase, atp-binding, phosphorylation, nucleotide-binding, alternative splicing, wnt signaling pathway, serine/threonine kinase
Biological sourceHOMO SAPIENS (HUMAN)
Cellular locationCytoplasm: Q9Y6M4
Total number of polymer chains1
Total formula weight39179.32
Authors
Primary citationBunkoczi, G.,Salah, E.,Rellos, P.,Das, S.,Fedorov, O.,Savitsky, P.,Debreczeni, J.E.,Gileadi, O.,Sundstrom, M.,Edwards, A.,Arrowsmith, C.,Weigelt, J.,von Delft, F.,Knapp, S.
Inhibitor Binding by Casein Kinases
To be Published,
Experimental method
X-RAY DIFFRACTION (1.3 Å)
Structure validation

218500

PDB entries from 2024-04-17

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