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2FQI

dual binding modes of a novel series of DHODH inhibitors

Summary for 2FQI
Entry DOI10.2210/pdb2fqi/pdb
Related2BXV 2FPT 2FPV 2FPY
DescriptorDihydroorotate dehydrogenase, mitochondrial, SULFATE ION, ACETATE ION, ... (7 entities in total)
Functional Keywordsprotein inhibitor complex, oxidoreductase
Biological sourceHomo sapiens (human)
Cellular locationMitochondrion inner membrane; Single-pass membrane protein: Q02127
Total number of polymer chains1
Total formula weight44665.07
Authors
Baumgartner, R.,Leban, J. (deposition date: 2006-01-18, release date: 2007-01-23, Last modification date: 2023-08-30)
Primary citationBaumgartner, R.,Walloschek, M.,Kralik, M.,Gotschlich, A.,Tasler, S.,Mies, J.,Leban, J.
Dual binding mode of a novel series of DHODH inhibitors.
J.Med.Chem., 49:1239-1247, 2006
Cited by
PubMed: 16480261
DOI: 10.1021/jm0506975
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.95 Å)
Structure validation

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