2E0A
Crystal structure of human pyruvate dehydrogenase kinase 4 in complex with AMPPNP
Summary for 2E0A
Entry DOI | 10.2210/pdb2e0a/pdb |
Descriptor | Pyruvate dehydrogenase kinase isozyme 4, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... (4 entities in total) |
Functional Keywords | pdk4, kinase, atp-binding, structural genomics, nppsfa, national project on protein structural and functional analyses, riken structural genomics/proteomics initiative, rsgi, transferase |
Biological source | Homo sapiens (human) |
Cellular location | Mitochondrion matrix: Q16654 |
Total number of polymer chains | 2 |
Total formula weight | 90602.99 |
Authors | Kukimoto-Niino, M.,Tokmakov, A.,Terada, T.,Shiromizu, I.,Kawamoto, M.,Matsusue, T.,Shirouzu, M.,Yokoyama, S.,RIKEN Structural Genomics/Proteomics Initiative (RSGI) (deposition date: 2006-10-03, release date: 2007-10-09, Last modification date: 2023-10-25) |
Primary citation | Kukimoto-Niino, M.,Tokmakov, A.,Terada, T.,Ohbayashi, N.,Fujimoto, T.,Gomi, S.,Shiromizu, I.,Kawamoto, M.,Matsusue, T.,Shirouzu, M.,Yokoyama, S. Inhibitor-bound structures of human pyruvate dehydrogenase kinase 4. Acta Crystallogr.,Sect.D, 67:763-773, 2011 Cited by PubMed: 21904029DOI: 10.1107/S090744491102405X PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.86 Å) |
Structure validation
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