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2AWZ

Hepatitis C Virus NS5b RNA Polymerase in complex with a covalent inhibitor (5h)

2AWZ の概要
エントリーDOI10.2210/pdb2awz/pdb
関連するPDBエントリー2AX0 2AX1
分子名称Genome polyprotein, SULFATE ION, 5R-(4-BROMOPHENYLMETHYL)-3-(BENZENESULFONYLAMINO)-4-OXO-2-THIONOTHIAZOLIDINE, ... (4 entities in total)
機能のキーワードhcv, ns5b, polymerase, fingers, thumb, palm, transferase
由来する生物種Hepatitis C virus
細胞内の位置Core protein p21: Host endoplasmic reticulum membrane; Single-pass membrane protein. Core protein p19: Virion (By similarity). Envelope glycoprotein E1: Virion membrane; Single-pass type I membrane protein (Potential). Envelope glycoprotein E2: Virion membrane; Single-pass type I membrane protein (Potential). p7: Host endoplasmic reticulum membrane; Multi-pass membrane protein (By similarity). Protease NS2-3: Host endoplasmic reticulum membrane; Multi-pass membrane protein (Potential). Serine protease NS3: Host endoplasmic reticulum membrane; Peripheral membrane protein (By similarity). Non-structural protein 4A: Host endoplasmic reticulum membrane; Single-pass type I membrane protein (Potential). Non-structural protein 4B: Host endoplasmic reticulum membrane; Multi-pass membrane protein (By similarity). Non-structural protein 5A: Host endoplasmic reticulum membrane; Peripheral membrane protein (By similarity). RNA-directed RNA polymerase: Host endoplasmic reticulum membrane; Single-pass type I membrane protein (Potential): P26663
タンパク質・核酸の鎖数2
化学式量合計130767.28
構造登録者
主引用文献Powers, J.P.,Piper, D.E.,Li, Y.,Mayorga, V.,Anzola, J.,Chen, J.M.,Jaen, J.C.,Lee, G.,Liu, J.,Peterson, M.G.,Tonn, G.R.,Ye, Q.,Walker, N.P.,Wang, Z.
SAR and Mode of Action of Novel Non-Nucleoside Inhibitors of Hepatitis C NS5b RNA Polymerase.
J.Med.Chem., 49:1034-1046, 2006
Cited by
PubMed: 16451069
DOI: 10.1021/jm050859x
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (2.15 Å)
構造検証レポート
Validation report summary of 2awz
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-03-27に公開中

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