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1W22

Crystal structure of inhibited human HDAC8

Summary for 1W22
Entry DOI10.2210/pdb1w22/pdb
Related1T64 1T67 1T69 1VKG
DescriptorHISTONE DEACETYLASE 8, ZINC ION, POTASSIUM ION, ... (5 entities in total)
Functional Keywordshydroxamic acid, chromatin, deacetylation, hdac, hydrolase, nuclear protein, repressor
Biological sourceHOMO SAPIENS
Cellular locationNucleus: Q9BY41
Total number of polymer chains2
Total formula weight84671.06
Authors
Vannini, A.,Volpari, C.,Caroli Casavola, E.,Di Marco, S. (deposition date: 2004-06-25, release date: 2004-09-24, Last modification date: 2023-12-13)
Primary citationVannini, A.,Volpari, C.,Filocamo, G.,Caroli Casavola, E.,Brunetti, M.,Renzoni, D.,Chakravarty, P.,Paolini, C.,De Francesco, R.,Gallinari, P.,Steinckuhler, C.,Di Marco, S.
Crystal Structure of a Eukaryotic Zn-Dependent Histone Deacetylase,Human Hdac8,Complexed with a Hydroxamic Acid Inhibitor
Proc.Natl.Acad.Sci.USA, 101:15064-, 2004
Cited by
PubMed: 15477595
DOI: 10.1073/PNAS.0404603101
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.5 Å)
Structure validation

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