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1CPU

SUBSITE MAPPING OF THE ACTIVE SITE OF HUMAN PANCREATIC ALPHA-AMYLASE USING SUBSTRATES, THE PHARMACOLOGICAL INHIBITOR ACARBOSE, AND AN ACTIVE SITE VARIANT

1CPU の概要
エントリーDOI10.2210/pdb1cpu/pdb
関連するBIRD辞書のPRD_IDPRD_900001
分子名称PROTEIN (ALPHA-AMYLASE), 4-amino-4,6-dideoxy-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ... (8 entities in total)
機能のキーワードamylase, acarbose, glycosylation, mutagenesis, diabetes, catalysis, pancreatic, enzyme, human, hydrolase
由来する生物種Homo sapiens (human)
タンパク質・核酸の鎖数1
化学式量合計57071.82
構造登録者
Brayer, G.D.,Sidhu, G.,Maurus, R.,Rydberg, E.H.,Braun, C.,Wang, Y.,Nguyen, N.T.,Overall, C.M.,Withers, S.G. (登録日: 1999-06-07, 公開日: 1999-06-14, 最終更新日: 2023-12-27)
主引用文献Brayer, G.D.,Sidhu, G.,Maurus, R.,Rydberg, E.H.,Braun, C.,Wang, Y.,Nguyen, N.T.,Overall, C.M.,Withers, S.G.
Subsite mapping of the human pancreatic alpha-amylase active site through structural, kinetic, and mutagenesis techniques.
Biochemistry, 39:4778-4791, 2000
Cited by
PubMed: 10769135
DOI: 10.1021/bi9921182
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (2 Å)
構造検証レポート
Validation report summary of 1cpu
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-03-27に公開中

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