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1C2K

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES

Summary for 1C2K
Entry DOI10.2210/pdb1c2k/pdb
Related1C1N 1C1O 1C1P 1C1Q 1C1R 1C1S 1C1T 1C1U 1C1V 1C1W 1C2D 1C2F 1C2G 1C2H 1C2I 1C2J 1C2L 1C2M
DescriptorTRYPSIN, CALCIUM ION, CHLORIDE ION, ... (6 entities in total)
Functional Keywordszn(ii)-mediated serine protease inhibitors, ph dependence, zn(ii) affinity stucture-based drug design, serine protease/inhibitor, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
Biological sourceBos taurus (cattle)
Cellular locationSecreted, extracellular space: P00760
Total number of polymer chains1
Total formula weight23691.82
Authors
Katz, B.A.,Luong, C. (deposition date: 1999-07-21, release date: 2000-07-26, Last modification date: 2023-12-27)
Primary citationKatz, B.A.,Clark, J.M.,Finer-Moore, J.S.,Jenkins, T.E.,Johnson, C.R.,Ross, M.J.,Luong, C.,Moore, W.R.,Stroud, R.M.
Design of potent selective zinc-mediated serine protease inhibitors.
Nature, 391:608-612, 1998
Cited by
PubMed: 9468142
DOI: 10.1038/35422
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.65 Å)
Structure validation

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