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8TCG
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BU of 8tcg by Molmil
Integrin alpha-v beta-6 in complex with minibinder B6_BP_dslf
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Integrin alpha-V heavy chain, ...
Authors:Campbell, M.G, Fernandez, A, Roy, A, Kraft, J, Baker, D.
Deposit date:2023-06-30
Release date:2023-09-27
Method:ELECTRON MICROSCOPY (3.4 Å)
Cite:De novo design of highly selective miniprotein inhibitors of integrins alpha v beta 6 and alpha v beta 8.
Nat Commun, 14, 2023
8TCF
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BU of 8tcf by Molmil
Integrin alpha-v beta-8 in complex with minibinder B8_BP_dsulf
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Campbell, M.G, Fernandez, A, Roy, A, Kraft, J, Baker, D.
Deposit date:2023-06-30
Release date:2023-09-27
Method:ELECTRON MICROSCOPY (2.9 Å)
Cite:De novo design of highly selective miniprotein inhibitors of integrins alpha v beta 6 and alpha v beta 8.
Nat Commun, 14, 2023
8T2U
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BU of 8t2u by Molmil
Cryo-EM Structures of Full-length Integrin alphaIIbbeta3 in Native Lipids complexed with Eptifibatide
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Adair, B, Xiong, J.P, Yeager, M, Arnaout, M.A.
Deposit date:2023-06-06
Release date:2023-07-26
Method:ELECTRON MICROSCOPY (3.1 Å)
Cite:Cryo-EM structures of full-length integrin alpha IIb beta 3 in native lipids.
Nat Commun, 14, 2023
8T2V
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BU of 8t2v by Molmil
Cryo-EM Structures of Full-length Integrin alphaIIbbeta3 in Native Lipids
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Adair, B, Xiong, J.P, Yeager, M, Arnaout, M.A.
Deposit date:2023-06-06
Release date:2023-07-26
Method:ELECTRON MICROSCOPY (3.4 Å)
Cite:Cryo-EM structures of full-length integrin alpha IIb beta 3 in native lipids.
Nat Commun, 14, 2023
8GCE
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BU of 8gce by Molmil
The Extracellular Domain of Integrin AlphaIIbBeta3 in Intermediate State
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Huo, T, Wu, H, Wang, Z.
Deposit date:2023-03-01
Release date:2024-03-06
Method:ELECTRON MICROSCOPY (3.12 Å)
Cite:Full-length AlphaIIbBeta3 CryoEM structure reveals intact integrin initiate-activation intrinsic architecture
To Be Published
8GCD
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BU of 8gcd by Molmil
Full length Integrin AlphaIIbBeta3 in inactive state
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Huo, T, Wu, H, Wang, Z.
Deposit date:2023-03-01
Release date:2024-03-06
Method:ELECTRON MICROSCOPY (2.97 Å)
Cite:Full-length AlphaIIbBeta3 CryoEM structure reveals intact integrin initiate-activation intrinsic architecture
To Be Published
8IJ5
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BU of 8ij5 by Molmil
Cryo-EM structure of Integrin AVB3
Descriptor: Integrin alpha-V heavy chain, Integrin beta-3
Authors:Xi, Z, Cang, W, Yuanzhu, G.
Deposit date:2023-02-26
Release date:2024-02-28
Method:ELECTRON MICROSCOPY (3 Å)
Cite:cryo-EM Structure of Integrin AVB3
To Be Published
7Y1T
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BU of 7y1t by Molmil
Complex of integrin alphaV/beta8 and L-TGF-beta1 at a ratio of 1:2
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Duan, Z, Zhang, Z.
Deposit date:2022-06-08
Release date:2022-08-31
Last modified:2022-09-07
Method:ELECTRON MICROSCOPY (3.24 Å)
Cite:Specificity of TGF-beta 1 signal designated by LRRC33 and integrin alpha V beta 8.
Nat Commun, 13, 2022
7USM
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BU of 7usm by Molmil
Integrin alphaM/beta2 ectodomain
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Goldsmith, J.A, McLellan, J.S.
Deposit date:2022-04-25
Release date:2022-08-17
Last modified:2022-09-14
Method:ELECTRON MICROSCOPY (2.7 Å)
Cite:Structural basis for non-canonical integrin engagement by Bordetella adenylate cyclase toxin.
Cell Rep, 40, 2022
7USL
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BU of 7usl by Molmil
Integrin alphaM/beta2 ectodomain in complex with adenylate cyclase toxin RTX751 and M1F5 Fab
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Goldsmith, J.A, McLellan, J.S.
Deposit date:2022-04-25
Release date:2022-08-17
Last modified:2022-09-14
Method:ELECTRON MICROSCOPY (2.7 Å)
Cite:Structural basis for non-canonical integrin engagement by Bordetella adenylate cyclase toxin.
Cell Rep, 40, 2022
7UKP
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BU of 7ukp by Molmil
Integrin alaphIIBbeta3 complex with a gantofiban analog
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-04-01
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.80112982 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UKT
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BU of 7ukt by Molmil
Integrin alaphIIBbeta3 complex with BMS4.2
Descriptor: (1-{[(5S)-3-(4-carbamimidoylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}piperidin-4-yl)acetic acid, 10E5 Fab heavy chain, 10E5 Fab light chain, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-04-01
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.36994433 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UKO
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BU of 7uko by Molmil
Integrin alaphIIBbeta3 complex with sibrafiban (Mn)
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-04-01
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.604 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UK9
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BU of 7uk9 by Molmil
Integrin alaphIIBbeta3 complex with lamifiban (Mn)
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-31
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.60001969 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UJE
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BU of 7uje by Molmil
Integrin alaphIIBbeta3 complex with UR2922 in Mn2+
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-30
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.499968 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UJK
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BU of 7ujk by Molmil
Integrin alaphIIBbeta3 complex with lamifiban
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-30
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.43265581 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UH8
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BU of 7uh8 by Molmil
Integrin alaphIIBbeta3 complex with roxifiban (Mn/Ca)
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-25
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.750024 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UFH
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BU of 7ufh by Molmil
Integrin alaphIIBbeta3 complex with fradafiban (Mn/Ca)
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-22
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.99768162 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UE0
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BU of 7ue0 by Molmil
Integrin alaphIIBbeta3 complex with fradafiban
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-20
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.741962 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UDH
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BU of 7udh by Molmil
Integrin alaphIIBbeta3 complex with BMS4-3
Descriptor: (4-{[(5S)-3-(piperidin-4-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}piperazin-1-yl)acetic acid, 10E5 Fab heavy chain, 10E5 Fab light chain, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-19
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.99998844 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UDG
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BU of 7udg by Molmil
Integrin alaphIIBbeta3 complex with lotrafiban
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-19
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.800069 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UCY
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BU of 7ucy by Molmil
Integrin alaphIIBbeta3 complex with gantofiban
Descriptor: (4-{[(5R)-3-(4-carbamimidoylphenyl)-2-oxo-1,3-oxazolidin-5-yl]methyl}piperazin-1-yl)acetic acid, 10E5 Fab heavy chain, 10E5 Fab light chain, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-17
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.34996319 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7UBR
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BU of 7ubr by Molmil
Integrin alaphIIBbeta3 complex with GR144053
Descriptor: 10E5 Fab heavy chain, 10E5 Fab light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-15
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.04992747 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7U9V
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BU of 7u9v by Molmil
Integrin alaphIIBbeta3 complex with BMS4-1
Descriptor: (4-{[(5S)-3-(4-carbamimidoylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}piperazin-1-yl)acetic acid, 10E5 Fab heavy chain, 10E5 light chain, ...
Authors:Zhu, J, Lin, F.-Y, Zhu, J, Springer, T.A.
Deposit date:2022-03-11
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.25492167 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022
7U9F
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BU of 7u9f by Molmil
Integrin alaphIIBbeta3 complex with BMS compound 4 in Mn2+
Descriptor: (4-{[(5S)-3-{4-[(E)-imino(4-methylpiperazin-1-yl)methyl]phenyl}-4,5-dihydro-1,2-oxazol-5-yl]methyl}piperazin-1-yl)acetic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Lin, F.-Y, Zhu, J, Zhu, J, Springer, T.A.
Deposit date:2022-03-10
Release date:2022-08-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.70000529 Å)
Cite:A general chemical principle for creating closure-stabilizing integrin inhibitors.
Cell, 185, 2022

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