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4PF3
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4pf3
MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN WITH COMPUOND 37A
Descriptor:Mineralocorticoid receptor
Authors:Sogabe, S., Habuka, N.
Deposit date:2014-04-28
Release date:2014-11-26
Method:X-RAY DIFFRACTION (1.1 Å)
Cite:Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists
Bioorg.Med.Chem., 22, 2014
1YMT
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1ymt
MOUSE SF-1 LBD
Descriptor:Steroidogenic factor 1, Nuclear receptor 0B2
Authors:Krylova, I.N., Sablin, E.P., Moore, J., Xu, R.X., Waitt, G.M., Juzumiene, D., Bynum, J.M., Fletterick, R.J., Willson, T.M., Ingraham, H.A.
Deposit date:2005-01-21
Release date:2005-03-15
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.2 Å)
Cite:Structural analyses reveal phosphatidyl inositols as ligands for the NR5 orphan receptors SF-1 and LRH-1
Cell(Cambridge,Mass.), 120, 2005
3UP3
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3up3
NUCLEAR RECEPTOR DAF-12 FROM HOOKWORM ANCYLOSTOMA CEYLANICUM IN COMPLEX WITH (25S)-CHOLESTENOIC ACID
Descriptor:aceDAF-12, Nuclear receptor coactivator 2
Authors:Zhi, X., Zhou, X.E., Melcher, K., Motola, D.L., Gelmedin, V., Hawdon, J., Kliewer, S.A., Mangelsdorf, D.J., Xu, H.E.
Deposit date:2011-11-17
Release date:2011-12-14
Modification date:2012-02-29
Method:X-RAY DIFFRACTION (1.25 Å)
Cite:Structural Conservation of Ligand Binding Reveals a Bile Acid-like Signaling Pathway in Nematodes.
J.Biol.Chem., 287, 2012
1FCY
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1fcy
ISOTYPE SELECTIVITY OF THE HUMAN RETINOIC ACID NUCLEAR RECEPTOR HRAR: THE COMPLEX WITH THE RARBETA/GAMMA-SELECTIVE RETINOID CD564
Descriptor:RETINOIC ACID RECEPTOR GAMMA-1
Authors:Klaholz, B.P., Mitschler, A., Moras, D., Structural Proteomics in Europe (SPINE)
Deposit date:2000-07-19
Release date:2000-09-11
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.3 Å)
Cite:Structural basis for isotype selectivity of the human retinoic acid nuclear receptor.
J.Mol.Biol., 302, 2000
3B0T
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3b0t
HUMAN VDR LIGAND BINDING DOMAIN IN COMPLEX WITH MAXACALCITOL
Descriptor:Vitamin D3 receptor
Authors:Hishiki, A., Hashimoto, H., Sato, M., Shimizu, T.
Deposit date:2011-06-14
Release date:2011-08-10
Method:X-RAY DIFFRACTION (1.3 Å)
Cite:Human VDR ligand binding domain in complex with maxacalcitol
To be Published
3VHV
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3vhv
MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN WITH NON-STEROIDAL ANTAGONIST
Descriptor:Mineralocorticoid receptor
Authors:Sogabe, S., Habuka, N.
Deposit date:2011-09-07
Release date:2011-12-28
Method:X-RAY DIFFRACTION (1.35 Å)
Cite:Identification of Benzoxazin-3-one Derivatives as Novel, Potent, and Selective Nonsteroidal Mineralocorticoid Receptor Antagonists
J.Med.Chem., 54, 2011
3AZ3
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3az3
CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR
Descriptor:Vitamin D receptor
Authors:Itoh, S., Iijima, S.
Deposit date:2011-05-20
Release date:2011-11-02
Method:X-RAY DIFFRACTION (1.36 Å)
Cite:Novel nonsecosteroidal vitamin D(3) carboxylic acid analogs for osteoporosis, and SAR analysis.
Bioorg.Med.Chem., 19, 2011
1FCZ
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1fcz
ISOTYPE SELECTIVITY OF THE HUMAN RETINOIC ACID NUCLEAR RECEPTOR HRAR: THE COMPLEX WITH THE PANAGONIST RETINOID BMS181156
Descriptor:RETINOIC ACID RECEPTOR GAMMA-1/INHIBITOR COMPLEX
Authors:Klaholz, B.P., Mitschler, A., Moras, D., Structural Proteomics in Europe (SPINE)
Deposit date:2000-07-19
Release date:2000-09-11
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.38 Å)
Cite:Structural basis for isotype selectivity of the human retinoic acid nuclear receptor.
J.Mol.Biol., 302, 2000
1FD0
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1fd0
ISOTYPE SELECTIVITY OF THE HUMAN RETINOIC ACID NUCLEAR RECEPTOR HRAR: THE COMPLEX WITH THE RARGAMMA-SELECTIVE RETINOID SR11254
Descriptor:RETINOIC ACID RECEPTOR GAMMA-1/INHIBITOR COMPLEX
Authors:Klaholz, B.P., Moras, D., Structural Proteomics in Europe (SPINE)
Deposit date:2000-07-19
Release date:2002-09-27
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.38 Å)
Cite:C-H...O hydrogen bonds in the nuclear receptor RARgamma--a potential tool for drug selectivity.
Structure, 10, 2002
1IE9
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1ie9
CRYSTAL STRUCTURE OF THE NUCLEAR RECEPTOR FOR VITAMIN D LIGAND BINDING DOMAIN BOUND TO MC1288
Descriptor:VITAMIN D3 RECEPTOR
Authors:Tocchini-Valentini, G., Rochel, N., Wurtz, J.M., Mitschler, A., Moras, D.
Deposit date:2001-04-09
Release date:2001-05-16
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:Crystal structures of the vitamin D receptor complexed to superagonist 20-epi ligands.
Proc.Natl.Acad.Sci.USA, 98, 2001
1T7R
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1t7r
CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN IN COMPLEX WITH A FXXLF MOTIF
Descriptor:Androgen receptor, FxxLF motif peptide
Authors:Hur, E., Pfaff, S.J., Payne, E.S., Gron, H., Buehrer, B.M., Fletterick, R.J.
Deposit date:2004-05-10
Release date:2004-08-31
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:Recognition and accommodation at the androgen receptor coactivator binding interface.
Plos Biol., 2, 2004
3WFG
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3wfg
MINERALOCORTICOID RECEPTOR LIGAND-BINDING DOMAIN WITH COMPUOND 2E
Descriptor:Mineralocorticoid receptor
Authors:Sogabe, S., Habuka, N.
Deposit date:2013-07-19
Release date:2013-08-21
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:Design, synthesis, and structure-activity relationships of dihydrofuran-2-one and dihydropyrrol-2-one derivatives as novel benzoxazin-3-one-based minera-locorticoid receptor antagonists
Bioorg.Med.Chem., 2013
4OHA
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4oha
CRYSTAL STRUCTURE OF T877A-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Descriptor:Androgen receptor, co-regulator peptide
Authors:Liu, J.S., Hsu, C.L., Wu, W.G.
Deposit date:2014-01-17
Release date:2014-08-20
Modification date:2014-12-24
Method:X-RAY DIFFRACTION (1.42 Å)
Cite:Identification of a new androgen receptor (AR) co-regulator BUD31 and related peptides to suppress wild-type and mutated AR-mediated prostate cancer growth via peptide screening and X-ray structure analysis.
Mol Oncol, 8, 2014
3A40
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3a40
CRYSTAL STRUCTURE OF THE HUMAN VDR LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND 2ALPHA-METHYL-AMCR277B(C23R)
Descriptor:Vitamin D3 receptor
Authors:Sato, Y., Antony, P., Huet, T., Sigueiro, R., Rochel, N., Moras, D.
Deposit date:2009-06-25
Release date:2010-02-02
Modification date:2013-11-20
Method:X-RAY DIFFRACTION (1.45 Å)
Cite:Structure-function relationships and crystal structures of the vitamin D receptor bound 2 alpha-methyl-(20S,23S)- and 2 alpha-methyl-(20S,23R)-epoxymethano-1 alpha,25-dihydroxyvitamin D3
J.Med.Chem., 53, 2010
1SQN
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1sqn
PROGESTERONE RECEPTOR LIGAND BINDING DOMAIN WITH BOUND NORETHINDRONE
Descriptor:progesterone receptor
Authors:Williams, S.P., Madauss, K.P., Deng, J.-S., Austin, R.J.H., Lambert, M.H., McLay, I., Pritchard, J., Short, S.A., Stewart, E.L., Uings, I.J.
Deposit date:2004-03-19
Release date:2004-07-27
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.451 Å)
Cite:Progesterone receptor ligand binding pocket flexibility: crystal structures of the norethindrone and mometasone furoate complexes
J.Med.Chem., 47, 2004
1SR7
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1sr7
PROGESTERONE RECEPTOR HORMONE BINDING DOMAIN WITH BOUND MOMETASONE FUROATE
Descriptor:Progesterone receptor
Authors:Madauss, K.P., Deng, S.-J., Austin, R.J., Lambert, M.H., McLay, I., Pritchard, J., Short, S.A., Stewart, E.L., Uings, I.J., Williams, S.P.
Deposit date:2004-03-22
Release date:2004-06-22
Modification date:2011-07-13
Method:X-RAY DIFFRACTION (1.46 Å)
Cite:Progesterone receptor ligand binding pocket flexibility: crystal structures of the norethindrone and mometasone furoate complexes
J.Med.Chem., 47, 2004
1FCX
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1fcx
ISOTYPE SELECTIVITY OF THE HUMAN RETINOIC ACID NUCLEAR RECEPTOR HRAR: THE COMPLEX WITH THE RARGAMMA-SELECTIVE RETINOID BMS184394
Descriptor:RETINOIC ACID RECEPTOR GAMMA-1
Authors:Klaholz, B.P., Mitschler, A., Moras, D., Structural Proteomics in Europe (SPINE)
Deposit date:2000-07-19
Release date:2000-09-11
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.47 Å)
Cite:Structural basis for isotype selectivity of the human retinoic acid nuclear receptor.
J.Mol.Biol., 302, 2000
3CJW
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3cjw
CRYSTAL STRUCTURE OF THE HUMAN COUP-TFII LIGAND BINDING DOMAIN
Descriptor:Crystal structure of the human COUP-TFII ligand binding domain
Authors:Kruse, S.W., Reynolds, R., Vonrhein, C., Xu, H.E.
Deposit date:2008-03-14
Release date:2008-10-07
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.48 Å)
Cite:Identification of COUP-TFII Orphan Nuclear Receptor as a Retinoic Acid-Activated Receptor.
Plos Biol., 6, 2008
1NQ7
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1nq7
CHARACTERIZATION OF LIGANDS FOR THE ORPHAN NUCLEAR RECEPTOR RORBETA
Descriptor:NUCLEAR RECEPTOR ROR-BETA
Authors:Stehlin-Gaon, C., Willmann, D., Sanglier, S., Van Dorsselaer, A., Renaud, J.-P., Moras, D., Schuele, R.
Deposit date:2003-01-21
Release date:2003-09-23
Modification date:2008-12-23
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:All-trans retinoic acid is a ligand for the orphan nuclear receptor RORbeta
Nat.Struct.Biol., 10, 2003
1YP0
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1yp0
STRUCTURE OF THE STEROIDOGENIC FACTOR-1 LIGAND BINDING DOMAIN BOUND TO PHOSPHOLIPID AND A SHP PEPTIDE MOTIF
Descriptor:nuclear receptor subfamily 5, group A, member 1, Nuclear receptor subfamily 0, group B, member 2
Authors:Li, Y., Choi, M., Cavey, G., Daugherty, J., Suino, K., Kovach, A., Bingham, N., Kliewer, S., Xu, H.
Deposit date:2005-01-28
Release date:2005-04-19
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Crystallographic identification and functional characterization of phospholipids as ligands for the orphan nuclear receptor steroidogenic factor-1.
Mol.Cell, 17, 2005
2AX6
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2ax6
CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN T877A MUTANT IN COMPLEX WITH HYDROXYFLUTAMIDE
Descriptor:Androgen receptor
Authors:Bohl, C.E., Miller, D.D., Chen, J., Bell, C.E., Dalton, J.T.
Deposit date:2005-09-03
Release date:2005-09-20
Modification date:2009-02-24
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Structural Basis for Accommodation of Nonsteroidal Ligands in the Androgen Receptor
J.Biol.Chem., 280, 2005
3AZ1
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3az1
CRYSTAL STRUCTURE ANALYSIS OF VITAMIN D RECEPTOR
Descriptor:Vitamin D3 receptor
Authors:Itoh, S., Iijima, S.
Deposit date:2011-05-20
Release date:2011-11-02
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Novel nonsecosteroidal vitamin D(3) carboxylic acid analogs for osteoporosis, and SAR analysis.
Bioorg.Med.Chem., 19, 2011
3MNP
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3mnp
CRYSTAL STRUCTURE OF THE AGONIST FORM OF MOUSE GLUCOCORTICOID RECEPTOR STABILIZED BY (A611V, V708A, E711G) MUTATIONS AT 1.50A
Descriptor:Glucocorticoid receptor, Nuclear receptor coactivator 2 protein
Authors:Schoch, G.A., Seitz, T., Benz, J., Banner, D., Stihle, M., D'Arcy, B., Thoma, R., Sterner, R., Hennig, M., Ruf, A.
Deposit date:2010-04-22
Release date:2010-09-15
Modification date:2011-01-19
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Enhancing the stability and solubility of the glucocorticoid receptor ligand-binding domain by high-throughput library screening.
J.Mol.Biol., 403, 2010
3OLL
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3oll
CRYSTAL STRUCTURE OF PHOSPHORYLATED ESTROGEN RECEPTOR BETA LIGAND BINDING DOMAIN
Descriptor:Estrogen receptor beta, Nuclear receptor coactivator 1
Authors:Moecklinghoff, S., Rose, R., Ottmann, C., Brunsveld, L.
Deposit date:2010-08-26
Release date:2010-11-17
Modification date:2010-12-08
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Synthesis and crystal structure of a phosphorylated estrogen receptor ligand binding domain.
Chembiochem, 11, 2010
3VTC
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3vtc
CRYSTAL STRUCTURE OF RAT VITAMIN D RECEPTOR BOUND TO A PARTIAL AGONIST 26-ADAMANTYL-23-YNE-19-NORVITAMMIN D ADTK3
Descriptor:Vitamin D3 receptor, COACTIVATOR PEPTIDE DRIP
Authors:Nakabayashi, M., Kudo, T., Tokiwa, H., Makishima, M., Yamada, S., Ikura, T., Ito, N.
Deposit date:2012-05-26
Release date:2013-06-12
Modification date:2014-05-14
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Combination of Triple Bond and Adamantane Ring on the Vitamin D Side Chain Produced Partial Agonists for Vitamin D Receptor.
J.Med.Chem., 2014
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entries available on 2015-07-01
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