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2ILM
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Factor Inhibiting HIF-1 Alpha D201A Mutant in Complex with FE(II), Alpha-Ketoglutarate and HIF-1 Alpha 35mer
分子名称: 2-OXOGLUTARIC ACID, BICARBONATE ION, FE (II) ION, ...
著者Mcdonough, M.A, Schofield, C.J.
登録日2006-10-03
公開日2007-08-14
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Evidence that two enzyme-derived histidine ligands are sufficient for iron binding and catalysis by factor inhibiting HIF (FIH).
J.Biol.Chem., 283, 2008
5JWP
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BU of 5jwp by Molmil
Crystal structure of human FIH D201E variant in complex with Zn, alpha-ketoglutarate, and HIF1 alpha peptide.
分子名称: 2-OXOGLUTARIC ACID, GLYCEROL, Hypoxia-inducible factor 1-alpha, ...
著者Taabazuing, C.Y, Garman, S.C, Eron, S, Knapp, M.J.
登録日2016-05-12
公開日2016-11-23
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The facial triad in the alpha-ketoglutarate dependent oxygenase FIH: A role for sterics in linking substrate binding to O2 activation.
J.Inorg.Biochem., 166, 2016
1H2L
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Factor Inhibiting HIF-1 alpha in complex with HIF-1 alpha fragment peptide
分子名称: 2-OXOGLUTARIC ACID, FACTOR INHIBITING HIF1, FE (II) ION, ...
著者Elkins, J.M, Hewitson, K.S, McNeill, L.A, Schlemminger, I, Seibel, J.F, Schofield, C.J.
登録日2002-08-12
公開日2002-11-28
最終更新日2018-02-21
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Structure of Factor-Inhibiting Hypoxia-Inducible Factor (Hif) Reveals Mechanism of Oxidative Modification of Hif-1Alpha
J.Biol.Chem., 278, 2003
1H2M
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Factor Inhibiting HIF-1 alpha in complex with HIF-1 alpha fragment peptide
分子名称: FACTOR INHIBITING HIF1, HYPOXIA-INDUCIBLE FACTOR 1 ALPHA, N-OXALYLGLYCINE, ...
著者Elkins, J.M, Hewitson, K.S, McNeill, L.A, Schlemminger, I, Seibel, J.F, Schofield, C.J.
登録日2002-08-12
公開日2002-11-28
最終更新日2018-02-21
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structure of Factor-Inhibiting Hypoxia-Inducible Factor (Hif) Reveals Mechanism of Oxidative Modification of Hif-1Alpha
J.Biol.Chem., 278, 2003
1H2K
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BU of 1h2k by Molmil
Factor Inhibiting HIF-1 alpha in complex with HIF-1 alpha fragment peptide
分子名称: FACTOR INHIBITING HIF1, FE (II) ION, HYPOXIA-INDUCIBLE FACTOR 1 ALPHA, ...
著者Elkins, J.M, Hewitson, K.S, McNeill, L.A, Schlemminger, I, Seibel, J.F, Schofield, C.J.
登録日2002-08-12
公開日2002-11-28
最終更新日2018-02-21
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structure of Factor-Inhibiting Hypoxia-Inducible Factor (Hif) Reveals Mechanism of Oxidative Modification of Hif-1Alpha
J.Biol.Chem., 278, 2003
7LVS
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BU of 7lvs by Molmil
The CBP TAZ1 Domain in Complex with a CITED2-HIF-1-Alpha Fusion Peptide
分子名称: Cbp/p300-interacting transactivator 2,Hypoxia-inducible factor 1-alpha, Histone lysine acetyltransferase CREBBP, ZINC ION
著者Appling, F.D, Berlow, R.B, Stanfield, R.L, Dyson, H.J, Wright, P.E.
登録日2021-02-26
公開日2021-07-28
最終更新日2021-12-15
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献The molecular basis of allostery in a facilitated dissociation process.
Structure, 29, 2021
7QGS
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Crystal structure of p300 CH1 domain in complex with CITIF (a CITED2-HIF-1alpha hybrid)
分子名称: Cbp/p300-interacting transactivator 2,Hypoxia-inducible factor 1-alpha, Histone acetyltransferase, ZINC ION
著者Hegedus, Z, Wilson, A.J, Edwards, T.A.
登録日2021-12-10
公開日2022-05-11
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Understanding p300-transcription factor interactions using sequence variation and hybridization.
Rsc Chem Biol, 3, 2022
1L8C
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STRUCTURAL BASIS FOR HIF-1ALPHA/CBP RECOGNITION IN THE CELLULAR HYPOXIC RESPONSE
分子名称: CREB-binding protein, Hypoxia-inducible factor 1 alpha, ZINC ION
著者Dames, S.A, Martinez-Yamout, M, De Guzman, R.N, Dyson, H.J, Wright, P.E.
登録日2002-03-19
公開日2002-04-10
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Structural basis for Hif-1 alpha /CBP recognition in the cellular hypoxic response.
Proc.Natl.Acad.Sci.USA, 99, 2002
1L3E
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BU of 1l3e by Molmil
NMR Structures of the HIF-1alpha CTAD/p300 CH1 Complex
分子名称: ZINC ION, hypoxia inducible factor-1 alpha subunit, p300 protein
著者Freedman, S.J, Sun, Z.J, Poy, F, Kung, A.L, Livingston, D.M, Wagner, G, Eck, M.J.
登録日2002-02-26
公開日2002-04-24
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Structural basis for recruitment of CBP/p300 by hypoxia-inducible factor-1 alpha.
Proc.Natl.Acad.Sci.USA, 99, 2002

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件を2024-04-17に公開中

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