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-Structure paper
Title | Complexes of HIV-1 reverse transcriptase with inhibitors of the HEPT series reveal conformational changes relevant to the design of potent non-nucleoside inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 39, Page 1589-1600, Year 1996 |
Publish date | Mar 16, 1996 (structure data deposition date) |
Authors | Hopkins, A.L. / Ren, J. / Esnouf, R.M. / Willcox, B.E. / Jones, E.Y. / Ross, C. / Miyasaka, T. / Walker, R.T. / Tanaka, H. / Stammers, D.K. / Stuart, D.I. |
External links | J. Med. Chem. / PubMed:8648598 |
Methods | X-ray diffraction |
Resolution | 2.55 Å |
Structure data | PDB-1rt1: PDB-1rt2: |
Chemicals | ChemComp-MKC: ChemComp-HOH: ChemComp-TNK: |
Source |
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Keywords | NUCLEOTIDYLTRANSFERASE / HIV-1 REVERSE TRANSCRIPTASE |