+Search query
-Structure paper
Title | Development of small molecule inhibitors of natural killer group 2D receptor (NKG2D). |
---|---|
Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 96, Page 129492-129492, Year 2023 |
Publish date | Apr 8, 2023 (structure data deposition date) |
Authors | Wang, J. / Nakafuku, K.M. / Ziff, J. / Gelin, C.F. / Gholami, H. / Thompson, A.A. / Karpowich, N.K. / Limon, L. / Coate, H.R. / Damm-Ganamet, K.L. ...Wang, J. / Nakafuku, K.M. / Ziff, J. / Gelin, C.F. / Gholami, H. / Thompson, A.A. / Karpowich, N.K. / Limon, L. / Coate, H.R. / Damm-Ganamet, K.L. / Shih, A.Y. / Grant, J.C. / Cote, M. / Mak, P.A. / Pascual, H.A. / Rives, M.L. / Edwards, J.P. / Venable, J.D. / Venkatesan, H. / Shi, Z. / Allen, S.J. / Sharma, S. / Kung, P.P. / Shireman, B.T. |
External links | Bioorg. Med. Chem. Lett. / PubMed:37778428 |
Methods | X-ray diffraction |
Resolution | 1.36 - 1.43 Å |
Structure data | PDB-8se5: PDB-8se6: |
Chemicals | ChemComp-PGE: ChemComp-PEG: ChemComp-ZW7: ChemComp-HOH: ChemComp-ZWA: ChemComp-PG4: |
Source |
|
Keywords | IMMUNE SYSTEM/INHIBITOR / NKG2D / Immune System / IMMUNOSUPPRESSANT-INHIBITOR complex / IMMUNE SYSTEM-INHIBITOR complex / DEL / cryptic pocket / immunoreceptors / SIGNALING PROTEIN |