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-Structure paper
Title | Comparative Study of Adenosine Analogs as Inhibitors of Protein Arginine Methyltransferases and a Clostridioides difficile- Specific DNA Adenine Methyltransferase. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 18, Page 734-745, Year 2023 |
Publish date | Jan 9, 2023 (structure data deposition date) |
Authors | Zhou, J. / Deng, Y. / Iyamu, I.D. / Horton, J.R. / Yu, D. / Hajian, T. / Vedadi, M. / Rotili, D. / Mai, A. / Blumenthal, R.M. ...Zhou, J. / Deng, Y. / Iyamu, I.D. / Horton, J.R. / Yu, D. / Hajian, T. / Vedadi, M. / Rotili, D. / Mai, A. / Blumenthal, R.M. / Zhang, X. / Huang, R. / Cheng, X. |
External links | Acs Chem. Biol. / PubMed:37082867 |
Methods | X-ray diffraction |
Resolution | 2.59 - 2.74 Å |
Structure data | PDB-8fs1: PDB-8fs2: |
Chemicals | ChemComp-EDO: ChemComp-YB0: ChemComp-K: ChemComp-HOH: ChemComp-YB5: |
Source |
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Keywords | TRANSFERASE/DNA/INHIBITOR / DNA Adenine Methylation / PROTEIN-DNA COMPLEX / TRANSFERASE / DNA BINDING PROTEIN / TRANSFERASE-DNA-INHIBITOR complex |