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-Structure paper
Title | Redesign of Rifamycin Antibiotics to Overcome ADP-Ribosylation-Mediated Resistance. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 61, Page e202211498-e202211498, Year 2022 |
Publish date | Feb 22, 2022 (structure data deposition date) |
Authors | Lan, T. / Ganapathy, U.S. / Sharma, S. / Ahn, Y.M. / Zimmerman, M. / Molodtsov, V. / Hegde, P. / Gengenbacher, M. / Ebright, R.H. / Dartois, V. ...Lan, T. / Ganapathy, U.S. / Sharma, S. / Ahn, Y.M. / Zimmerman, M. / Molodtsov, V. / Hegde, P. / Gengenbacher, M. / Ebright, R.H. / Dartois, V. / Freundlich, J.S. / Dick, T. / Aldrich, C.C. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:36222275 |
Methods | X-ray diffraction |
Resolution | 3.87 Å |
Structure data | PDB-7u22: |
Chemicals | ChemComp-KYO: ChemComp-ZN: ChemComp-MG: |
Source |
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Keywords | ANTIBIOTIC / Transcription / inhibitor / rifabutin / transcription initiation / tuberculosis / MTB / Mycobacterium tuberculosis / Mycobacterium smegmatis |