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-Structure paper
Title | Discovery of Potent Selective Nonzinc Binding Autotaxin Inhibitor BIO-32546. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 12, Page 1124-1129, Year 2021 |
Publish date | Apr 9, 2021 (structure data deposition date) |
Authors | Ma, B. / Zhang, L. / Sun, L. / Xin, Z. / Kumaravel, G. / Marcotte, D. / Chodaparambil, J.V. / Wang, Q. / Wehr, A. / Jing, J. ...Ma, B. / Zhang, L. / Sun, L. / Xin, Z. / Kumaravel, G. / Marcotte, D. / Chodaparambil, J.V. / Wang, Q. / Wehr, A. / Jing, J. / Hong, V.S. / Wang, T. / Huang, C. / Shao, Z. / Mi, S. |
External links | Acs Med. Chem. Lett. / PubMed:34267882 |
Methods | X-ray diffraction |
Resolution | 2.3 Å |
Structure data | PDB-7mfh: |
Chemicals | ChemComp-ZF7: ChemComp-IOD: ChemComp-EDO: ChemComp-ZN: ChemComp-PEG: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE/INHIBITOR / hydrolase inhibitor / Autotaxin / HYDROLASE / HYDROLASE-INHIBITOR complex |