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-Structure paper
Title | Anti-obesity effects of GIPR antagonists alone and in combination with GLP-1R agonists in preclinical models. |
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Journal, issue, pages | Sci Transl Med, Vol. 10, Year 2018 |
Publish date | May 29, 2018 (structure data deposition date) |
Authors | Killion, E.A. / Wang, J. / Yie, J. / Shi, S.D. / Bates, D. / Min, X. / Komorowski, R. / Hager, T. / Deng, L. / Atangan, L. ...Killion, E.A. / Wang, J. / Yie, J. / Shi, S.D. / Bates, D. / Min, X. / Komorowski, R. / Hager, T. / Deng, L. / Atangan, L. / Lu, S.C. / Kurzeja, R.J.M. / Sivits, G. / Lin, J. / Chen, Q. / Wang, Z. / Thibault, S.A. / Abbott, C.M. / Meng, T. / Clavette, B. / Murawsky, C.M. / Foltz, I.N. / Rottman, J.B. / Hale, C. / Veniant, M.M. / Lloyd, D.J. |
External links | Sci Transl Med / PubMed:30567927 |
Methods | X-ray diffraction |
Resolution | 1.95 Å |
Structure data | PDB-6dkj: |
Chemicals | ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | SIGNALING PROTEIN / GPCR |