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-Structure paper
Title | Identification of a PDE4-Specific Pocket for the Design of Selective Inhibitors. |
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Journal, issue, pages | Biochemistry, Vol. 57, Page 4518-4525, Year 2018 |
Publish date | Jul 14, 2017 (structure data deposition date) |
Authors | Feng, X. / Wang, H. / Ye, M. / Xu, X.T. / Xu, Y. / Yang, W. / Zhang, H.T. / Song, G. / Ke, H. |
External links | Biochemistry / PubMed:29975048 |
Methods | X-ray diffraction |
Resolution | 1.6 - 1.8 Å |
Structure data | PDB-5wh5: PDB-5wh6: |
Chemicals | ChemComp-R91: ChemComp-ZN: ChemComp-MG: ChemComp-HOH: ChemComp-AKJ: |
Source |
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Keywords | Hydrolase/Hydrolase Inhibitor / Phosphodiesterase / inhibitors / Hydrolase-Hydrolase Inhibitor complex / inhibitor Zl-n-91 / PDE4D-S91 complex |