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-Structure paper
Title | Bisubstrate Udp-Peptide Conjugates as Human O-Glcnac Transferase Inhibitors. |
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Journal, issue, pages | Biochem. J., Vol. 457, Page 497-, Year 2014 |
Publish date | Nov 5, 2013 (structure data deposition date) |
Authors | Borodkin, V.S. / Schimpl, M. / Gundogdu, M. / Rafie, K. / Dorfmueller, H.C. / Robinson, D.A. / Van Aalten, D.M. |
External links | Biochem. J. / PubMed:24256146 |
Methods | X-ray diffraction |
Resolution | 3.15 Å |
Structure data | PDB-4cdr: |
Chemicals | ChemComp-SO4: ChemComp-UDP: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX / INVERTING GT-B ENZYME / BI-SUBSTRATE ANALOG INHIBITOR |