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-Structure paper
Title | Structure-guided inhibitor design expands the scope of analog-sensitive kinase technology. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 8, Page 1931-1938, Year 2013 |
Publish date | Jun 27, 2013 (structure data deposition date) |
Authors | Zhang, C. / Lopez, M.S. / Dar, A.C. / Ladow, E. / Finkbeiner, S. / Yun, C.H. / Eck, M.J. / Shokat, K.M. |
External links | Acs Chem. Biol. / PubMed:23841803 |
Methods | X-ray diffraction |
Resolution | 2.41 - 2.84 Å |
Structure data | PDB-4lgg: PDB-4lgh: |
Chemicals | ChemComp-VGG: ChemComp-HOH: ChemComp-0JN: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Kinase Domain / TRANSFERASE-TRANSFERASE INHIBITOR complex |