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-Structure paper
Title | Discovery of Novel Jak2-Stat Pathway Inhibitors with Extended Residence Time on Target. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 23, Page 3105-, Year 2013 |
Publish date | Feb 11, 2013 (structure data deposition date) |
Authors | Guan, H. / Lamb, M.L. / Peng, B. / Huang, S. / Degrace, N. / Read, J. / Hussain, S. / Wu, J. / Rivard, C. / Alimzhanov, M. ...Guan, H. / Lamb, M.L. / Peng, B. / Huang, S. / Degrace, N. / Read, J. / Hussain, S. / Wu, J. / Rivard, C. / Alimzhanov, M. / Bebernitz, G. / Bell, K. / Ye, M. / Zinda, M. / Ioannidis, S. |
External links | Bioorg. Med. Chem. Lett. / PubMed:23562594 |
Methods | X-ray diffraction |
Resolution | 2.51 Å |
Structure data | PDB-3zmm: |
Chemicals | ChemComp-F9J: ChemComp-ACE: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE |