タイトル | Structure-activity analysis of aging and reactivation of human butyrylcholinesterase inhibited by analogues of tabun. |
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ジャーナル・号・ページ | Biochem. J., Vol. 421, Page 97-106, Year 2009 |
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掲載日 | 2009年5月11日 (構造データの登録日) |
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著者 | Carletti, E. / Aurbek, N. / Gillon, E. / Loiodice, M. / Nicolet, Y. / Fontecilla-Camps, J.C. / Masson, P. / Thiermann, H. / Nachon, F. / Worek, F. |
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リンク | Biochem. J. / PubMed:19368529 |
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手法 | X線回折 |
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解像度 | 2 - 3.1 Å |
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構造データ | PDB-2wid: NONAGED FORM OF HUMAN BUTYRYLCHOLINESTERASE INHIBITED BY TABUN ANALOGUE TA1 手法: X-RAY DIFFRACTION / 解像度: 2.3 Å PDB-2wif: AGED FORM OF HUMAN BUTYRYLCHOLINESTERASE INHIBITED BY TABUN ANALOGUE TA1 手法: X-RAY DIFFRACTION / 解像度: 2.25 Å PDB-2wig: NONAGED FORM OF HUMAN BUTYRYLCHOLINESTERASE INHIBITED BY TABUN ANALOGUE TA4 手法: X-RAY DIFFRACTION / 解像度: 2.15 Å PDB-2wij: NONAGED FORM OF HUMAN BUTYRYLCHOLINESTERASE INHIBITED BY TABUN ANALOGUE TA5 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-2wik: NONAGED FORM OF HUMAN BUTYRYLCHOLINESTERASE INHIBITED BY TABUN ANALOGUE TA6 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-2wil: AGED FORM OF HUMAN BUTYRYLCHOLINESTERASE INHIBITED BY TABUN ANALOGUE TA5 手法: X-RAY DIFFRACTION / 解像度: 3.1 Å PDB-2wsl: Aged Form of Human Butyrylcholinesterase Inhibited by Tabun Analogue TA4 手法: X-RAY DIFFRACTION / 解像度: 2.0 Å |
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化合物 | |
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由来 | ![](img/tx_human.gif) homo sapiens (ヒト)
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キーワード | HYDROLASE (加水分解酵素) / AGING (老化) / INHIBITION (酵素阻害剤) / POLYMORPHISM / GLYCOPROTEIN (糖タンパク質) / SERINE ESTERASE / DISEASE MUTATION / TABUN / BUTYRYLCHOLINESTERASE |
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