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-Structure paper
Title | Benzothiazole based inhibitors of p38alpha MAP kinase. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 18, Page 1874-1879, Year 2008 |
Publish date | Feb 1, 2008 (structure data deposition date) |
Authors | Liu, C. / Lin, J. / Pitt, S. / Zhang, R.F. / Sack, J.S. / Kiefer, S.E. / Kish, K. / Doweyko, A.M. / Zhang, H. / Marathe, P.H. ...Liu, C. / Lin, J. / Pitt, S. / Zhang, R.F. / Sack, J.S. / Kiefer, S.E. / Kish, K. / Doweyko, A.M. / Zhang, H. / Marathe, P.H. / Trzaskos, J. / Mckinnon, M. / Dodd, J.H. / Barrish, J.C. / Schieven, G.L. / Leftheris, K. |
External links | Bioorg. Med. Chem. Lett. / PubMed:18296051 |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | PDB-3c5u: |
Chemicals | ChemComp-P41: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / SERINE/THREONINE-PROTEIN KINASE / KINASE / P38 MAP KINASE / Alternative splicing / ATP-binding / Cytoplasm / Nucleotide-binding / Nucleus / Phosphoprotein |