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-Structure paper
Title | Binding of the second generation non-nucleoside inhibitor S-1153 to HIV-1 reverse transcriptase involves extensive main chain hydrogen bonding. |
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Journal, issue, pages | J. Biol. Chem., Vol. 275, Page 14316-14320, Year 2000 |
Publish date | Mar 27, 2000 (structure data deposition date) |
Authors | Ren, J. / Nichols, C. / Bird, L.E. / Fujiwara, T. / Sugimoto, H. / Stuart, D.I. / Stammers, D.K. |
External links | J. Biol. Chem. / PubMed:10799511 |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | PDB-1ep4: |
Chemicals | ChemComp-S11: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / HIV-1 reverse transcriptase / AIDS / non-nucleoside inhibitor / S-1153 / drug design |