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1ITO
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BU of 1ito by Molmil
Crystal Structure Analysis of Bovine Spleen Cathepsin B-E64c complex
Descriptor: Cathepsin B, N-[1-HYDROXYCARBOXYETHYL-CARBONYL]LEUCYLAMINO-2-METHYL-BUTANE
Authors:Yamamoto, A, Tomoo, T, Matsugi, K, Hara, T, In, Y, Murata, M, Kitamura, K, Ishida, T.
Deposit date:2002-01-19
Release date:2003-01-19
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.286 Å)
Cite:Structural basis for development of cathepsin B-specific noncovalent-type inhibitor: crystal structure of cathepsin B-E64c complex
BIOCHIM.BIOPHYS.ACTA, 1597, 2002
5AWX
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BU of 5awx by Molmil
Crystal structure of Human PTPRZ D1 domain
Descriptor: BROMIDE ION, Receptor-type tyrosine-protein phosphatase zeta
Authors:Sugawara, H.
Deposit date:2015-07-10
Release date:2016-02-17
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.86 Å)
Cite:Small-molecule inhibition of PTPRZ reduces tumor growth in a rat model of glioblastoma
Sci Rep, 6, 2016
6AHS
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BU of 6ahs by Molmil
Mouse Kallikrein 7 in complex with imidazolinylindole derivative
Descriptor: 1-[(2-chlorophenyl)sulfonyl]-5-methyl-3-[(4R)-2-methyl-4,5-dihydro-1H-imidazol-4-yl]-1H-indole, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
Authors:Sugawara, H.
Deposit date:2018-08-20
Release date:2019-01-02
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Discovery and structure-activity relationship of imidazolinylindole derivatives as kallikrein 7 inhibitors.
Bioorg. Med. Chem. Lett., 29, 2019
5ZFI
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BU of 5zfi by Molmil
Mouse kallikrein 7 in complex with 6-benzyl-1,4-diazepan-7-one derivative
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 2-[(3Z,6R)-6-[(2,6-dichlorophenyl)methyl]-3-(dimethylhydrazinylidene)-7-oxo-1,4-diazepan-1-yl]-N-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]acetamide, Kallikrein-7
Authors:Sugawara, H.
Deposit date:2018-03-06
Release date:2018-06-27
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Structure-based drug design to overcome species differences in kallikrein 7 inhibition of 1,3,6-trisubstituted 1,4-diazepan-7-ones.
Bioorg. Med. Chem., 26, 2018
5ZFH
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BU of 5zfh by Molmil
Mouse Kallikrein 7
Descriptor: Kallikrein-7
Authors:Sugawara, H.
Deposit date:2018-03-06
Release date:2018-06-27
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (1.93 Å)
Cite:Structure-based drug design to overcome species differences in kallikrein 7 inhibition of 1,3,6-trisubstituted 1,4-diazepan-7-ones.
Bioorg. Med. Chem., 26, 2018
5H08
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BU of 5h08 by Molmil
Human PTPRZ D1 domain complexed with NAZ2329
Descriptor: 3-{[2-Ethoxy-5-(trifluoromethyl)benzyl]sulfanyl}-N-(phenylsulfonyl)thiophene-2-carboxamide, Receptor-type tyrosine-protein phosphatase zeta
Authors:Sugawara, H.
Deposit date:2016-10-04
Release date:2017-07-26
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.53 Å)
Cite:Targeting PTPRZ inhibits stem cell-like properties and tumorigenicity in glioblastoma cells
Sci Rep, 7, 2017
6J6U
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BU of 6j6u by Molmil
Rat PTPRZ D1-D2 domain
Descriptor: Receptor-type tyrosine-protein phosphatase zeta
Authors:Sugawara, H.
Deposit date:2019-01-15
Release date:2019-08-28
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (3.32 Å)
Cite:A head-to-toe dimerization has physiological relevance for ligand-induced inactivation of protein tyrosine receptor type Z.
J.Biol.Chem., 294, 2019

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