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5V2L
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BU of 5v2l by Molmil
Mevalonate diphosphate mediated ATP binding mechanism of the mevalonate diphosphate decarboxylase from Enterococcus faecalis
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, Mevalonate diphosphate decarboxylase, PHOSPHATE ION
Authors:Stauffacher, C.V, Chen, C.-L.
Deposit date:2017-03-05
Release date:2017-10-18
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Mevalonate 5-diphosphate mediates ATP binding to the mevalonate diphosphate decarboxylase from the bacterial pathogen Enterococcus faecalis.
J. Biol. Chem., 292, 2017
5V2M
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BU of 5v2m by Molmil
Mevalonate diphosphate mediated ATP binding mechanism of the mevalonate diphosphate decarboxylase from Enterococcus faecalis
Descriptor: Mevalonate diphosphate decarboxylase, SULFATE ION
Authors:Stauffacher, C.V, Chen, C.-L.
Deposit date:2017-03-05
Release date:2017-10-18
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.989 Å)
Cite:Mevalonate 5-diphosphate mediates ATP binding to the mevalonate diphosphate decarboxylase from the bacterial pathogen Enterococcus faecalis.
J. Biol. Chem., 292, 2017
1XWW
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BU of 1xww by Molmil
Crystal Structure of Human B-form Low Molecular Weight Phosphotyrosyl Phosphatase at 1.6 Angstrom Resolution
Descriptor: GLYCEROL, Low molecular weight phosphotyrosine protein phosphatase, SULFATE ION
Authors:Stauffacher, C.V, Zabell, A.P.R.
Deposit date:2004-11-02
Release date:2005-11-01
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (1.63 Å)
Cite:Crystal structure of the human B-form low molecular weight phosphotyrosyl phosphatase at 1.6-A resolution.
J.Biol.Chem., 281, 2006
4I4B
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BU of 4i4b by Molmil
HMG-CoA Reductase from Pseudomonas mevalonii complexed with NAD and intermediate hemiacetal form of HMG-CoA
Descriptor: (3R,5R,9R,19R,21S)-1-[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-hydroxy-3-(phosphonooxy)tetrahydrofuran-2-yl]-3,5,9,21-tetrahydroxy-8,8,21-trimethyl-10,14-dioxo-19-sulfanyl-2,4,6-trioxa-18-thia-11,15-diaza-3,5-diphosphatricosan-23-oic acid 3,5-dioxide, (3S)-3-hydroxy-3-methyl-5-sulfanylpentanoic acid, 3-hydroxy-3-methylglutaryl-coenzyme A reductase, ...
Authors:Stauffacher, C.V, Steussy, C.N, Critchelow, C.J, Schmidt, T, Min, J, Wrensford, L.V, Burgner, J.W, Rodwell, V.W.
Deposit date:2012-11-27
Release date:2013-07-17
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:A Novel Role for Coenzyme A during Hydride Transfer in 3-Hydroxy-3-methylglutaryl-coenzyme A Reductase.
Biochemistry, 52, 2013
6E2S
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BU of 6e2s by Molmil
apo form of MDDEF with buffer exchange
Descriptor: Mevalonate diphosphate decarboxylase, SULFATE ION
Authors:Stauffacher, C.V, Chen, C.-L.
Deposit date:2018-07-12
Release date:2020-01-15
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (1.791 Å)
Cite:Visualizing the enzyme mechanism of mevalonate diphosphate decarboxylase.
Nat Commun, 11, 2020
6E2T
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BU of 6e2t by Molmil
MDDEF in complex with MVAPP
Descriptor: (3R)-3-HYDROXY-5-{[(R)-HYDROXY(PHOSPHONOOXY)PHOSPHORYL]OXY}-3-METHYLPENTANOIC ACID, Mevalonate diphosphate decarboxylase
Authors:Stauffacher, C.V, Chen, C.-L.
Deposit date:2018-07-12
Release date:2020-01-15
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (1.692 Å)
Cite:Visualizing the enzyme mechanism of mevalonate diphosphate decarboxylase.
Nat Commun, 11, 2020
6E2U
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BU of 6e2u by Molmil
MDDEF in complex with MVAPP, AMPPCP and Magnesium
Descriptor: (3R)-3-HYDROXY-5-{[(R)-HYDROXY(PHOSPHONOOXY)PHOSPHORYL]OXY}-3-METHYLPENTANOIC ACID, MAGNESIUM ION, Mevalonate diphosphate decarboxylase, ...
Authors:Stauffacher, C.V, Chen, C.-L.
Deposit date:2018-07-12
Release date:2020-01-15
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.05 Å)
Cite:Visualizing the enzyme mechanism of mevalonate diphosphate decarboxylase.
Nat Commun, 11, 2020
6E2W
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BU of 6e2w by Molmil
MDDEF in complex with MVAPP, ADP, sulfate and cobalt
Descriptor: (3R)-3-HYDROXY-5-{[(R)-HYDROXY(PHOSPHONOOXY)PHOSPHORYL]OXY}-3-METHYLPENTANOIC ACID, ADENOSINE-5'-DIPHOSPHATE, COBALT (II) ION, ...
Authors:Stauffacher, C.V, Chen, C.-L.
Deposit date:2018-07-12
Release date:2020-01-15
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Visualizing the enzyme mechanism of mevalonate diphosphate decarboxylase.
Nat Commun, 11, 2020
6E2V
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BU of 6e2v by Molmil
MDDEF in complex with MVAPP, ADPBeF3 and magnesium
Descriptor: (3R)-3-HYDROXY-5-{[(R)-HYDROXY(PHOSPHONOOXY)PHOSPHORYL]OXY}-3-METHYLPENTANOIC ACID, ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, ...
Authors:Stauffacher, C.V, Chen, C.-L.
Deposit date:2018-07-12
Release date:2020-01-15
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Visualizing the enzyme mechanism of mevalonate diphosphate decarboxylase.
Nat Commun, 11, 2020
6E2Y
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BU of 6e2y by Molmil
MDDEF in complex with MVAPP, ADP, sulfate and cobalt. Anomalous data
Descriptor: (3R)-3-HYDROXY-5-{[(R)-HYDROXY(PHOSPHONOOXY)PHOSPHORYL]OXY}-3-METHYLPENTANOIC ACID, ADENOSINE-5'-DIPHOSPHATE, COBALT (II) ION, ...
Authors:Stauffacher, C.V, Chen, C.-L.
Deposit date:2018-07-12
Release date:2020-01-15
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.34 Å)
Cite:Visualizing the enzyme mechanism of mevalonate diphosphate decarboxylase.
Nat Commun, 11, 2020
1C0E
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BU of 1c0e by Molmil
Active Site S19A Mutant of Bovine Heart Phosphotyrosyl Phosphatase
Descriptor: PHOSPHATE ION, PROTEIN (TYROSINE PHOSPHATASE (ORTHOPHOSPHORIC MONOESTER PHOSPHOHYDROLASE))
Authors:Tabernero, L, Evans, B.N, Tishmack, P.A, Van Etten, R.L, Stauffacher, C.V.
Deposit date:1999-07-15
Release date:1999-09-28
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:The structure of the bovine protein tyrosine phosphatase dimer reveals a potential self-regulation mechanism.
Biochemistry, 38, 1999
8GDN
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BU of 8gdn by Molmil
Structure of PmHMGR bound to mevalonate, CoA and NAD.
Descriptor: (R)-MEVALONATE, 3-hydroxy-3-methylglutaryl-coenzyme A reductase, COENZYME A, ...
Authors:Purohit, V, Steussy, C.N, Stauffacher, C.V.
Deposit date:2023-03-06
Release date:2024-03-20
Method:X-RAY DIFFRACTION (1.99 Å)
Cite:pH-dependent reaction triggering in PmHMGR crystals for time-resolved crystallography.
Biophys.J., 123, 2024
8VLQ
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BU of 8vlq by Molmil
Structure of PmHMGR bound to mevalonate, CoA and NAD 5 minutes after reaction initiation at pH 9
Descriptor: (R)-MEVALONATE, (R)-mevaldehyde, 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, ...
Authors:Purohit, V, Steussy, C.N, Stauffacher, C.V.
Deposit date:2024-01-12
Release date:2024-03-20
Method:X-RAY DIFFRACTION (2.07 Å)
Cite:pH-dependent reaction triggering in PmHMGR crystals for time-resolved crystallography.
Biophys.J., 123, 2024
8SZ6
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BU of 8sz6 by Molmil
PmHMGR bound to mevaldehyde and CoA
Descriptor: (3R)-3,5,5-trihydroxy-3-methylpentanoic acid, 3-hydroxy-3-methylglutaryl-coenzyme A reductase, Mevaldyl-Coenzyme A, ...
Authors:Purohit, V, Stauffacher, C.V, Steussy, C.N.
Deposit date:2023-05-27
Release date:2024-03-20
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:pH-dependent reaction triggering in PmHMGR crystals for time-resolved crystallography.
Biophys.J., 123, 2024
5JNP
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BU of 5jnp by Molmil
Crystal structure of a rice (Oryza Sativa) cellulose synthase plant conserved region (P-CR)
Descriptor: CITRATE ANION, GLYCEROL, PHOSPHATE ION, ...
Authors:Rushton, P.S, Olek, A.T, Makowski, L, Badger, J, Steussy, C.N, Carpita, N.C, Stauffacher, C.V.
Deposit date:2016-04-30
Release date:2016-12-28
Last modified:2019-12-04
Method:X-RAY DIFFRACTION (2.404 Å)
Cite:Rice Cellulose SynthaseA8 Plant-Conserved Region Is a Coiled-Coil at the Catalytic Core Entrance.
Plant Physiol., 173, 2017
3N8I
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BU of 3n8i by Molmil
Crystal structure of the A isoform of human cytoplasmic protein tyrosine phosphatase (HCPTP-A) in complex with 1-naphtylacetic acid
Descriptor: Low molecular weight phosphotyrosine protein phosphatase, NAPHTHALEN-1-YL-ACETIC ACID
Authors:Homan, K.T, Balasubramaniam, D, Stauffacher, C.V.
Deposit date:2010-05-28
Release date:2011-12-07
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Structural Characterization of a Secondary Binding Site on Low Molecular Weight Protein Tyrosine Phosphatases
To be Published
1D2A
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BU of 1d2a by Molmil
CRYSTAL STRUCTURE OF A YEAST LOW MOLECULAR WEIGHT PROTEIN TYROSINE PHOSPHATASE (LTP1) COMPLEXED WITH THE ACTIVATOR ADENINE
Descriptor: ADENINE, CHLORIDE ION, PHOSPHATE ION, ...
Authors:Wang, S, Stauffacher, C.V, Van Etten, R.L.
Deposit date:1999-09-22
Release date:2000-03-01
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Structural and mechanistic basis for the activation of a low-molecular weight protein tyrosine phosphatase by adenine.
Biochemistry, 39, 2000
7M3H
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BU of 7m3h by Molmil
Targeting Enterococcus faecalis HMG-CoA reductase with a novel non-statin inhibitor
Descriptor: 5-[(4-butylphenyl)sulfamoyl]-2-hydroxybenzoic acid, CALCIUM ION, Hydroxymethylglutaryl-CoA reductase, ...
Authors:Bose, S, Steussy, C.N, Stauffacher, C.V.
Deposit date:2021-03-18
Release date:2022-09-21
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (1.27 Å)
Cite:Targeting Enterococcus faecalis HMG-CoA reductase with a novel non-statin inhibitor
To Be Published
2HDB
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BU of 2hdb by Molmil
HMG-CoA synthase from Enterococcus faecalis. Mutation alanine 110 to glycine
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, HMG-CoA synthase, SULFATE ION
Authors:Steussy, C.N, Sutherlin, A, Stauffacher, C.V.
Deposit date:2006-06-20
Release date:2007-03-20
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:A structural limitation on enzyme activity: the case of HMG-CoA synthase.
Biochemistry, 45, 2006
2I88
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BU of 2i88 by Molmil
Crystal structure of the Channel-forming Domain of Colicin E1
Descriptor: Colicin-E1
Authors:Elkins, P, Bunker, A, Cramer, W.A, Stauffacher, C.V.
Deposit date:2006-09-01
Release date:2006-09-26
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:A mechanism for toxin insertion into membranes is suggested by the crystal structure of the channel-forming domain of colicin E1
Structure, 5, 1997
1X9E
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BU of 1x9e by Molmil
Crystal structure of HMG-CoA synthase from Enterococcus faecalis
Descriptor: HMG-CoA synthase, SULFATE ION
Authors:Steussy, C.N, Vartia, A.A, Burgner II, J.W, Sutherlin, A, Rodwell, V.W, Stauffacher, C.V.
Deposit date:2004-08-20
Release date:2005-11-01
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:X-ray Crystal Structures of HMG-CoA Synthase from Enterococcus faecalis and a Complex with Its Second Substrate/Inhibitor Acetoacetyl-CoA
Biochemistry, 44, 2005
7M1Z
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BU of 7m1z by Molmil
Targeting Enterococcus faecalis HMG-CoA reductase with a novel non-statin inhibitor
Descriptor: (R)-MEVALONATE, 3-HYDROXY-3-METHYLGLUTARYL-COENZYME A, ACETATE ION, ...
Authors:Bose, S, Steussy, C.N, Stauffacher, C.V.
Deposit date:2021-03-15
Release date:2022-09-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.27 Å)
Cite:Targeting Enterococcus faecalis HMG-CoA reductase with a non-statin inhibitor
Nat Commun, 2023
1D1P
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BU of 1d1p by Molmil
CRYSTAL STRUCTURE OF A YEAST LOW MOLECULAR WEIGHT PROTEIN TYROSINE PHOSPHATASE (LTP1)
Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, TYROSINE PHOSPHATASE
Authors:Wang, S, Tabernero, L, Zhang, M, Harms, E, Van Etten, R.L, Stauffacher, C.V.
Deposit date:1999-09-20
Release date:2000-03-08
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Crystal structures of a low-molecular weight protein tyrosine phosphatase from Saccharomyces cerevisiae and its complex with the substrate p-nitrophenyl phosphate.
Biochemistry, 39, 2000
1CK1
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BU of 1ck1 by Molmil
STRUCTURE OF STAPHYLOCOCCAL ENTEROTOXIN C3
Descriptor: PROTEIN (ENTEROTOXIN TYPE C-3), ZINC ION
Authors:Chi, Y.-I, Bohach, G.A, Stauffacher, C.V.
Deposit date:1999-04-26
Release date:2002-07-10
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Zinc-mediated dimerization and its effect on activity and conformation of staphylococcal enterotoxin type C.
J.Biol.Chem., 277, 2002
1DG9
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BU of 1dg9 by Molmil
CRYSTAL STRUCTURE OF BOVINE LOW MOLECULAR WEIGHT PTPASE COMPLEXED WITH HEPES
Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, TYROSINE PHOSPHATASE
Authors:Zhang, M, Zhou, M, Van Etten, R.L, Stauffacher, C.V.
Deposit date:1999-11-23
Release date:1999-12-08
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Crystal structure of bovine low molecular weight phosphotyrosyl phosphatase complexed with the transition state analog vanadate.
Biochemistry, 36, 1997

 

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